Relugolix is used to treat advanced prostate cancer (cancer that begins in the prostate [a male reproductive gland]) in adult men. Relugolix is in a class of medications called gonadotropin-releasing hormone (GnRH) receptor antagonists. It works by decreasing the amount of testosterone (a male hormone) produced by the body. This may slow or stop the spread of prostate cancer cells that need testosterone to grow.
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Prostate cancer is a slow-growing cancer that originates in the prostate gland and can spread to other parts of the body.
Rexilo 120mg Tablet contains Relugolix, an Anti-androgen medication used to treat prostate cancer in adult males.
Symptoms of prostate cancer include troubled urination, blood in urine, frequent night-time urination, blood in semen, bone pain, unintentional weight loss, pain while sitting, and erectile dysfunction. During treatment with Rexilo 120mg Tablet, your doctor may conduct blood tests to monitor changes in your blood.
While taking Rexilo 120mg Tablet, avoid excessive direct exposure to sunlight or UV light. Inform your doctor about any existing liver or heart issues, as well as diabetes, before starting the medication. Rexilo 120mg Tablet is not suitable for use in women, including pregnant or breastfeeding women.
This medication is also not recommended for children and adolescents under 18 years of age. Common side effects of Rexilo 120mg Tablet include skin rash, breast swelling or tenderness, weakness, loss of appetite, dizziness, sleepiness, and nausea. If any of these symptoms worsen over time, contact your doctor.
Avoid consumption of alcohol while taking Rexilo 120mg Tablet.
Rexilo 120mg Tablet is not recommended for use in pregnant women. Patients and their partners should use birth control while taking Rexilo 120mg Tablet and for 130 days after stopping the treatment. Consult your doctor before taking it.
Rexilo 120mg Tablet is not recommended for use in breastfeeding women. Consult your doctor before taking it.
Do not drive or operate any machines if you feel sleepy after taking Rexilo 120mg Tablet.
No dosage adjustment of Rexilo 120 is necessary for patients with kidney impairment. Consult your doctor before taking it.
Rexilo 120mg Tablet should be used with caution in patients with liver problems. Consult your doctor before taking it.
Relugolix tablets work by decreasing the amount of testosterone (a male hormone) produced by the body. This may slow or stop the spread of prostate cancer cells that need testosterone to grow.
Take Rexilo 120mg Tablet as advised by your physician. Swallow with a glass of water and do not chew or crush it. Your doctor will decide the correct dose and duration of Rexilo 120mg Tablet treatment for you depending on your age, body weight, and disease condition. Do not stop taking Rexilo 120mg Tablet unless your doctor advises you to stop.
Calutide 50 mg Tablet is a non-steroidal anti-cancer medicine used in men along with other specific agents for the treatment of prostate cancer. This medicine is not recommended for use in females, children, and adolescents.
Rexilo 120mg Tablet is an anti-androgen medication that exerts its pharmacological effects by inhibiting the action of androgens, which are male sex hormones responsible for the growth and development of the prostate gland. Prostate cancer cells depend on androgens to grow and spread, so by blocking the androgen receptors, Rexilo 120mg Tablet prevents the cancer cells from receiving the signals that promote their growth.
By inhibiting the androgen receptors, Rexilo 120mg Tablet slows down the growth of prostate cancer cells and reduces their ability to spread to other parts of the body. This action helps in controlling the progression of prostate cancer and alleviating the symptoms associated with it.
The drug is usually taken orally as a tablet, and its effects are specific to androgen receptors in the prostate gland, sparing other tissues from similar inhibition. Rexilo 120mg Tablet works alongside other treatments for prostate cancer to improve outcomes and quality of life for patients with this condition. However, it is essential to follow the prescribed dosage and consult the doctor regularly for monitoring and adjusting the treatment plan as necessary.
When taking Relugolix, it is important to be cautious about potential drug interactions. Some medications may affect the blood levels of Relugolix, leading to increased side effects or reduced effectiveness. In particular,Relugolix can cause a serious heart problem, and the risk may be higher when combined with certain other medications used for various conditions.
To minimize the risk of interactions, certain drugs should not be taken within 6 hours after you take Relugolix. It is crucial to carefully follow your doctor's instructions regarding the scheduling of all your medications. Always inform your doctor about all the medications you are taking, including prescription and over-the-counter medicines, vitamins, and herbal products, to avoid any harmful interactions. Your doctor can assess the potential interactions and adjust your treatment plan accordingly to ensure your safety and optimal treatment outcomes.
Before starting relugolix, it's crucial to consider the following:
It's important to communicate with your doctor about any pre-existing conditions or potential risks before using this medication. Following your doctor's advice and using appropriate birth control methods can help ensure the safe and effective use of relugolix.
This drug has shown embryo-fetal lethality in animal studies at maternal exposures 0.3 times the human exposure at the recommended dose of 120 mg daily, based on AUC. There are no controlled data on human pregnancy.
The US FDA has not assigned a specific pregnancy category for this drug. Safety and efficacy during pregnancy have not been established. Patients should be aware that this drug can cause fetal harm and loss of pregnancy based on animal studies and its mechanism of action. Therefore, it is important to advise patients of the potential risk to the fetus.
This drug may also impair fertility. Males with female partners of reproductive potential should use effective contraception during therapy and for at least 2 weeks after the last dose.
Regarding lactation, it is unknown whether this drug is excreted into human milk. In animal studies, the drug and its metabolites were present in the milk of lactating animals, with concentrations up to 10-fold higher than in plasma at 2 hours post-dose after a single oral dose of 30 mg/kg on post-partum day 14. The effects in nursing infants are unknown, and there is no specific recommendation for use during breastfeeding.
Because the drug is approximately 68 to 71% bound to plasma proteins and has a half-life of about 25 hours, it may accumulate in the infant if excreted into breast milk. Further research is needed to understand the potential risks to nursing infants.
Keep this medication in the container it came in, tightly closed, and out of reach of children. Store it at room temperature and away from excess heat and moisture (not in the bathroom). Do not remove the desiccant (small packet included with medication to absorb moisture).
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